Bulletin of the Chemical Society of Japan
Online ISSN : 1348-0634
Print ISSN : 0009-2673
ISSN-L : 0009-2673
α,β-Epoxy Sulfoxides as Useful Intermediates in Organic Synthesis. III. A Novel Synthesis of α-Amino Ketones and α-Amino Aldehydes by Aminolysis of α,β-Epoxy Sulfoxides
Tsuyoshi SatohYouhei KanekoKiichi SakataKoji Yamakawa
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1986 Volume 59 Issue 2 Pages 457-463

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Abstract

Aminolysis of α,β-epoxy sulfoxides, easily prepared from 1-chloroalkyl phenyl sulfoxides or chloromethyl phenyl sulfoxide and carbonyl compounds, with alkyl- or arylamines afforded α-amino ketones or α-amino aldehydes in good yields. Treatment of thus obtained α-arylamino ketones with weak Lewis acid led to 2,3-disubstituted indoles.

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