YAKUGAKU ZASSHI
Online ISSN : 1347-5231
Print ISSN : 0031-6903
ISSN-L : 0031-6903
総説
実用的イミダゾリン合成法の開発とその展開
村井 健一
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ジャーナル フリー

2010 年 130 巻 8 号 p. 1011-1016

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抄録
  This review describes the first method to prepare imidazolines from aldehydes and 1,2-diamines by condensation and successive oxidation using NBS in one-pot operation. The reaction proceeds under mild conditions and can be applied to various aromatic and aliphatic aldehydes and 1,2-diamines. The utility of this method is also demonstrated in the total synthesis of spongotine A and the preparation of a newly designed organocatalyst, C3-symmetric trisimidazoline 7.
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© 2010 by the PHARMACEUTICAL SOCIETY OF JAPAN
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