1962 年 82 巻 11 号 p. 1558-1560
Condensation of methyl ethyl ketone and 5-nitro-2-furfural diacetate afforded 1, 5-bis(5-nitro-2-furyl)-2-methyl-3-pentadienone (I) and 3-methyl-4-(5-nitro-2-furyl)-3-buten-2-one (II). By the reaction of these compounds with aminoguanidine, their amidinohydrazone hydrochlorides were purified. Heating of the amidinohydrazone of (I) in organic solvent, in the presence of alkaline substance, gave 3-amino-6-[1-methyl-2-(5-nitro-2-furyl)vinyl]-as-triazine. Antibacterial activity of these compounds was examined and interesting results were obtained.