1964 年 84 巻 4 号 p. 372-373
Optically active N2-phthaloylaspartimide was synthesized from pharmacological interest. The optically active N2-phthaloylasparagine, obtained by resolution of racemic compound with brucine, was found to undergo dehydrative cyclization by the action of acetyl chloride under a mild condition to form the optically active N2-phthaloylaspartimide.