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Abstracts of Annual meeting of Japanese Society for the Study of Xenobiotics
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19th Annual meeting of the Japanese Society for the Study of Xenobiotics
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17th Annual meeting of JSSX
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30th JSSX Annual meeting
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26th JSSX Annual meeting
25th JSSX Annual meeting
24th JSSX Annual meeting
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19th Annual meeting of the Japanese Society for the Study of Xenobiotics
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[volume title in Japanese]
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17th Annual meeting of JSSX
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Distinguished Lectures
Molecular Mechanism of Drug Metabolizing Enzymes — Glucuronosyltransferase —
Takashi Iyanagi
Session ID: D1
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.1.0
CONFERENCE PROCEEDINGS
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(782K)
Computer Simulation of Cellular Processes and its applications to Biotechnology
[in Japanese]
Session ID: D2
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.2.0
CONFERENCE PROCEEDINGS
FREE ACCESS
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(1127K)
Rapid Identification of Novel Genes by Hybrid-Ribozyme Libraries
Kazunari TAIRA
Session ID: D3
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.3.0
CONFERENCE PROCEEDINGS
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(863K)
Symposium 1A
REGULATION OF HUMAN
CYP3A
GENES
Tetsuya SAITO, Shunsuke IWANO, Keiko MATSUMURA, Yoshiki TAKAHASHI, Tet ...
Session ID: 21S1A-01
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.4.0
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(774K)
Molecular Mechanism of human CYP3A4 induction and construction of its validation system
Kiyoshi NAGATA, Tomonari TAKADA, Takahiro OHKUBO, Yoko NAGAI, Masayuki ...
Session ID: 21S1A-02
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.5.0
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(649K)
REGULATION MECHANISM FOR CELLULAR LOCALIZATION AND EXPRESSION OF CONSTITUTIVE ACTIVE RECEPTOR (CAR)
Kaoru KOBAYASHI, Tatsuya SUEYOSHI, Rick MOORE, Masahiko NEGISHI
Session ID: 21S1A-03
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.6.0
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(739K)
Mechansim of CYP2B2 gene regulation in the Qdj:SD rat, a mutant strain which lacks PB-mediated response to CYP2B2 induction
H. Matsunaga, R. Matsumoto, Y. Shirabe, K. Oguri, H. Yamada
Session ID: 21S1A-04
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.7.0
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(685K)
Structural organization and characterization of the regulatory element of the human carboxylesterase gene
Masakiyo HOSOKAWA, Natsuko WATANABE, Yumiko YAGINUMA, Misato DAIMON, E ...
Session ID: 21S1A-05
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.8.0
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(862K)
REGULATION OF CYP2D EXPRESSION: A NOVEL TRANSCRIPTIONAL REGULATION SYSTEM OF CYP2D4 EXPRESSION IN THE BRAIN
Dai Mizuno, Yoshiki Takahashi, Toyoko Hiroi, Susumu Imaoka, Tetsuya Ka ...
Session ID: 21S1A-06
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.9.0
CONFERENCE PROCEEDINGS
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(669K)
EVALUATION OF GENE INDUCTION OF DRUG-METABOLIZING ENZYMES IN HUMAN HEPATOCYTES
Shinsaku NAITO, Masuhiro NISHIMURA, Satoshi SUZUKI, Tetsuo SATOH
Session ID: 22S1A-01
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.10.0
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(814K)
EVALUATION OF CYP-INDUCTION AND DRUG METABOLISM USING HUMAN HEPATOCYTES
Kaoru SHIMADA
Session ID: 22S1A-02
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.11.0
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(882K)
HORMONAL REGULATION OF THE EXPRESSION OF MOUSE CYP3A ISOFORMS
Tsutomu SAKUMA, Yusuke ENDO, Misae MASHINO, Nobuo NEMOTO
Session ID: 22S1A-03
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.12.0
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(811K)
Symposium 1B
Relationship between Single Nucleotide Polymorphism of CYP2D6 and Enzymatic Functions: Focusing on the N-terminal Region
Daisuke TSUZUKI, Yukie OKUDA, Shigeo YAMAMOTO, Hiroyuki KATAOKA, Shizu ...
Session ID: 21S1B-01
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.13.0
CONFERENCE PROCEEDINGS
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(791K)
Genetic polymorphisms of human
CYP2A6
gene and interindividual differences in nicotine metabolism
Miki NAKAJIMA, Ryoko YOSHIDA, Jun-Tack KWON, Yukio KUROIWA, Tsuyoshi Y ...
Session ID: 21S1B-02
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.14.0
CONFERENCE PROCEEDINGS
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(700K)
GENETIC POLYMORPHISMS IN DRUG-ADMINISTERED JAPANESE PATIENTS
Shogo Ozawa
Session ID: 21S1B-03
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.15.0
CONFERENCE PROCEEDINGS
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(706K)
GENETIC POLYMORPHISMS AND FUNCTIONAL CHARACTERIZATION OF THE HUMAN OATP-C GENE
Ichiro IEIRI, Yohei NISHIZATO, Hiroshi SUZUKI, Miyuki KIMURA, Kiyoshi ...
Session ID: 21S1B-04
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.16.0
CONFERENCE PROCEEDINGS
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(726K)
CLINICAL USE OF SNPs INFORMATION
Junichi AZUMA, Masako OHNO, Tsuyoshi FUKUDA
Session ID: 21S1B-05
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.17.0
CONFERENCE PROCEEDINGS
FREE ACCESS
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(810K)
MDR1
Genotyping for Individualization of Drug Therapy
T. Sakaeda, T. Nakamura, K. Okumura
Session ID: 21S1B-06
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.18.0
CONFERENCE PROCEEDINGS
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(767K)
Application of genotyping in clinical therapy: Medication for patients with bone marrow transfer
Noritaka ARIYOSHI, Michiko MIZUNO, Takashi SUZUKI, Kenji OKADA, Masahi ...
Session ID: 22S1B-01
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.19.0
CONFERENCE PROCEEDINGS
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(850K)
THE EFFECTS OF GENETIC POLYMORPHISMS, SMOKING AND OTHER FACTIORS ON THE METABOLISM AND EXTENT OF DRUG-INTERACTIONS OF FLUVOXAMINE
Hisakazu OHTANI, Chiharu MAEBARA, Hideyo SUGAHARA, Matsuko TANAKA, Nor ...
Session ID: 22S1B-02
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.20.0
CONFERENCE PROCEEDINGS
FREE ACCESS
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(757K)
Symposium 2
PHYSIOLOGICAL AND PHARMACOLOGICAL RELEVANCE OF OCTN TRANSPORTERS
Ikumi TAMAI, Yoshimichi SAI, Akira TSUJI
Session ID: 20S2-01
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.21.0
CONFERENCE PROCEEDINGS
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(960K)
STRUCTURAL AND FUNCTIONAL ANALYSES OF RENAL DRUG TRANSPORTERS AND THEIR CLINICAL IMPLICATIONS
Hideyuki SAITO, Satohiro MASUDA, Hideyuki MOTOHASHI, Yumiko URAKAMI, Y ...
Session ID: 20S2-02
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.22.0
CONFERENCE PROCEEDINGS
FREE ACCESS
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(952K)
EXPRESSION OF ABC TRANSPORTER A AND G FAMILIES AT THE BRAIN BARRIER
Sumio Ohtsuki, Satoko Hori, Taro Suda, Azusa Sato, Yuki Watanabe, Mayu ...
Session ID: 20S2-03
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.23.0
CONFERENCE PROCEEDINGS
FREE ACCESS
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(759K)
HUMAN ABC TRANSPORTERS: FROM GENOMIC ANALYSIS TO DATABASE CONSTRUCTION, FUNCTIONAL SCREENING, AND DRUG MOLECULAR DESIGN
Toshihisa ISHIKAWA, Yoji IKEGAMI, Hikaru YABUUCHI, Masato KITAJIMA
Session ID: 20S2-04
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.24.0
CONFERENCE PROCEEDINGS
FREE ACCESS
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(815K)
The in vivo/in vitro extrapolation of the metabolic inhibition and induction in liver and the first pass metabolism in intestine for drugs
Motohiro Kato
Session ID: 20S2-05
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.25.0
CONFERENCE PROCEEDINGS
FREE ACCESS
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(744K)
SIGNIFICANCE OF IMPROVEMENT AND REGULATION OF INTESTINAL XENOBIOTIC ABSORPTION AND EXCRETION BASED ON TRANSPORT MECHANISM ACROSS EPITHELIA
Mikio TOMITA, Mayuko NAGIRA, Masahiro HAYASHI
Session ID: 20S2-06
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.26.0
CONFERENCE PROCEEDINGS
FREE ACCESS
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(956K)
QUANTITATIVE PREDICTION OF ORAL ABSORPTION OF DRUGS THAT ARE SUBSTRATES OF OLIGOPEPTIDE TRANSPORTER (PEPT1)
Rikako Shimizu, Tomomi Sukegawa, Kiyomi Ito, Yasuyuki Tsuda, Shuhei Ta ...
Session ID: 20S2-07
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.27.0
CONFERENCE PROCEEDINGS
FREE ACCESS
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(780K)
DRUG-DRUG INTERACTION CAUSED BY THE INHIBITION OF TRANSPORTER-MEDIATED HEPATIC UPTAKE
Yoshihisa SHITARA, Kazuya MAEDA, Tomoo ITOH, Hitoshi SATO, Albert P. L ...
Session ID: 20S2-08
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.28.0
CONFERENCE PROCEEDINGS
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(923K)
DDS technology to control the intracellular pharmacokinetics
Shinsaku Nakagawa
Session ID: 20S2-09
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.29.0
CONFERENCE PROCEEDINGS
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(958K)
Development of Multifunctional Vaccines through Optimization of In Vivo Disposition Characteristics and Intracellular Localization by Chemical Modification
Yasuomi Yamasaki, Takayuki Ohtsuki, Tomoko Ikenaga, Kohsuke Shakushiro ...
Session ID: 20S2-10
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.30.0
CONFERENCE PROCEEDINGS
FREE ACCESS
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(882K)
FUNCTIONAL CHARACTERIZATION OF SYSTEM L AMINO ACID TRANSPORTER(S) IN NEURAL CELLS: THE RELATIONSHIP WITH PHARMACOLOGICAL ACTIVITY OF GABAPENTIN
Takuya FUJITA, Miyuki WADA, Akira YAMAMOTO
Session ID: 20S2-11
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.31.0
CONFERENCE PROCEEDINGS
FREE ACCESS
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(806K)
ANTICOAGULANT THERAPY BASED ON GENETIC FACTORS AFFECTING PHARMACOKINETICS AND PHARMACODYNAMICS OF WARFARIN
Harumi TAKAHASHI, Toshitaka KASHIMA, Grant R WILKINSON, Ichiro IEIRI, ...
Session ID: 20S2-12
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.32.0
CONFERENCE PROCEEDINGS
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(894K)
PERSONALIZED MEDICINE BY THE SNP DETECTION
Masahiro HIRATSUKA, Yukinaga KISHIKAWA, Michinao MIZUGAKI
Session ID: 20S2-13
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.33.0
CONFERENCE PROCEEDINGS
FREE ACCESS
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(758K)
Symposium 3
View on Utilization of
In Silico
PK/ADME/TK Solution in Drug Discovery
[in Japanese]
Session ID: 20S3-01
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.34.0
CONFERENCE PROCEEDINGS
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(592K)
[title in Japanese]
[in Japanese]
Session ID: 20S3-02
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.35.0
CONFERENCE PROCEEDINGS
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(819K)
‘DRUGLIKE LIBRARY FOR DRUG DISCOVERY’
Noriaki Hirayama
Session ID: 20S3-03
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.36.0
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(758K)
THE AVAILABILITY OF
IN SILICO
ADME MODELS DURING LEAD OPTIMIZATION
Toshiyuki KUME, Tsunehiro HARADA
Session ID: 20S3-04
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.37.0
CONFERENCE PROCEEDINGS
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(962K)
ADME RESEARCH TOWARD VIRTUAL SCREENING
Shinji YAMASHITA
Session ID: 20S3-05
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.38.0
CONFERENCE PROCEEDINGS
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(903K)
QSAR ANALYSIS OF INTESTINAL MEMBRANE PERMEABILITY USING NOVEL INFORMATIC APPROACHES
Shin-ichi FUJIWARA, Fumiyoshi YAMASHITA, Mitsuru HASHIDA
Session ID: 20S3-06
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.39.0
CONFERENCE PROCEEDINGS
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(682K)
Information Technology in the Field of Drug Metabolism and Pharmacokinetics
Masato Kitajima, Jose Martin Ciloy, Kotaro Yuta
Session ID: 20S3-07
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.40.0
CONFERENCE PROCEEDINGS
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(560K)
In Silico
Predictive ADME Solutions and their Use to Support Decisions in Drug Discovery
Kevin Holme
Session ID: 20S3-08
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.41.0
CONFERENCE PROCEEDINGS
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(672K)
THE APPLICATION OF
IN SILICO
ADME TOOLS IN DRUG DISCOVERY
Mike Tarbit
Session ID: 20S3-09
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.42.0
CONFERENCE PROCEEDINGS
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(648K)
[title in Japanese]
Akira AKAMATSU
Session ID: 20S3-10
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.43.0
CONFERENCE PROCEEDINGS
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(809K)
TREND OF DRUG DISCOVERY BY SYSTEM BIOLOGY
Hirotugu WATABE
Session ID: 20S3-11
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.44.0
CONFERENCE PROCEEDINGS
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(272K)
Forum 2002
ROLE OF MASS BALANCE STUDY IN DRUG DEVELOPMENT
Yasuo OHNO
Session ID: F-1
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.45.0
CONFERENCE PROCEEDINGS
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(499K)
[title in Japanese]
[in Japanese]
Session ID: F-2
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.46.0
CONFERENCE PROCEEDINGS
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(793K)
MESURMENT OF NATURAL LEVEL OF
14
C WITH ACCELRATOR MASS SPECTROMETER
Hideyo NOGUCHI
Session ID: F-3
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.47.0
CONFERENCE PROCEEDINGS
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(602K)
INTERNAL DOSIMETRY BY ICRP
Hiroshi NOGUCHI
Session ID: F-5
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.49.0
CONFERENCE PROCEEDINGS
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(799K)
The Regulatory, Legal and Ethical Framework for Studies of Drug Metabolism and Pharmacokinetics in Human Volunteers in the West
Alan M Johnston
Session ID: F-6
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.50.0
CONFERENCE PROCEEDINGS
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(317K)
CLINICAL PHARMACOLOGICAL ASPECTS ON HUMAN MASS BALANCE STUDY
Kyoichi OHASHI
Session ID: F-7
Published: 2002
Released on J-STAGE: November 27, 2009
DOI
https://doi.org/10.14896/jssxmeeting.17.0.51.0
CONFERENCE PROCEEDINGS
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(583K)
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