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Abstracts of Annual meeting of Japanese Society for the Study of Xenobiotics
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19th Annual meeting of the Japanese Society for the Study of Xenobiotics
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17th Annual meeting of JSSX
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25th JSSX Annual meeting
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President's Lecture
TOWARD INTERNATIONALIZATION OF JSSX
Ken-ichi Inui
Session ID: PL
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.1.0
CONFERENCE PROCEEDINGS
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(395K)
Distinguished Lectures
SYSTEMS BIOLOGY OF MAMMALIAN CIRCADIAN CLOCKS
Hiroki Ueda
Session ID: DL-1
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.2.0
CONFERENCE PROCEEDINGS
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(403K)
CHEMICALLY REACTIVE METABOLITES IN DRUG DISCOVERY AND LEAD OPTIMIZATION
Thomas Allan Baillie
Session ID: DL-2
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.3.0
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(347K)
JSSX 25th Anniversary Symposium
Towards the Next Stage of DMPK Research by Integrating Uncovered Roles of Enzymes and Transporters - Challenges for Innovative Drug Discovery and Pharmacotherapy -
TARGETED RADIONUCLIDE THERAPY – PRACTICE OF TARGETING CONFIRMATIVE THERAPY, AN INDIVIDUALIZED IMAGE-BASED TREATMENT
Seigo Kinuya
Session ID: MS-1
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.4.0
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(482K)
MOLECULAR IMAGING ESPECIALLY PET - A USEFUL TOOL FOR IN VIVO MEASUREMENTS IN DRUG DEVELOPMENT
Bengt Langstrom
Session ID: MS-2
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.5.0
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(380K)
APPLICATION OF PHYSIOLOGICALLY BASED PHARMACOKINETIC(PBPK) MODELING AND CLEARANCE CONCEPT TO THE ANALYSIS OF TRANSPORTER-MEDIATED DISTRIBUTION AND CLEARANCE OF DRUGS IN HUMAN
Yuichi Sugiyama
Session ID: MS-3
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.6.0
CONFERENCE PROCEEDINGS
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(366K)
HUMAN DRUG METABOLITES AND INTERACTIONS MEDIATED POLYMORPHIC DRUG-METABOLIZING ENZYMES
Hiroshi Yamaza
Session ID: MS-4
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.7.0
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(367K)
PRECLINICAL STUDIES ON DRUG METABOLISM AND PHARMACOKINETICS IN STRATEGIC DRUG DISCOVERY FOR SUCCESSFUL DEVELOPMENT OF NEW DRUGS
Masato Chiba
Session ID: MS-5
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.8.0
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(367K)
SCIENTIFIC PERSPECTIVE ON CYP- AND TRANSPORTER- BASED DRUG-DRUG INTERACTIONS: IMPACT ON DRUG EXPOSURE/RESPONSE, LABELING AND CLINICAL DECISIONS
Shiew-Mei Huang
Session ID: MS-6
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.9.0
CONFERENCE PROCEEDINGS
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(381K)
Symposium 1
JSSX Symposium for the Success in Drug Development 2nd Symposium - PK/PD Based Functional Linkage for Drug Discovery and Development
PK/PD, BIOMARKER + MODEL-BASED DRUG DEVELOPMENT
WHERE TO START?
Ulrich Roth
Session ID: S1-1
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.10.0
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(362K)
MEDCHEM MEETS ADME
Atsushi Naganawa, Koji Yano, Yoshiyuki Yamaura, Soonih Kim
Session ID: S1-2
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.11.0
CONFERENCE PROCEEDINGS
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(387K)
ADME RESEARCH IN DRUG DEVELOPMENT OF ANTI-CANCER AGENTS
Kunihiro Yoshisue
Session ID: S1-3
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.12.0
CONFERENCE PROCEEDINGS
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(367K)
FORMULATION DESIGN AND PHARMACOKINETICS CONTROL
Kazuhiro Sako
Session ID: S1-4
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.13.0
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(367K)
COOPERATION OF DMPK AND TOX FOR DISCOVERY AND DEVELOPMENT OF SAFE DRUG
Takahiko Baba
Session ID: S1-5
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.14.0
CONFERENCE PROCEEDINGS
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(368K)
Symposium 2
Drug Metabolism Research in Asia: Orphan P450 enzymes, Natural Products, and Human Metabolite Formations
ROLES OF P450 1A AND 3A ENZYMES INVOLVED IN REACTIVE METABOLITE FORMATIONS
Hiroshi Yamazaki
Session ID: S2-1
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.15.0
CONFERENCE PROCEEDINGS
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(362K)
GENERATION OF HUMAN DRUG METABOLITES BY BACTERIAL CYTOCHROME P450 BM3 MUTANTS
Chul-Ho Yun
Session ID: S2-2
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.16.0
CONFERENCE PROCEEDINGS
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(387K)
ELUCIDATING THE FUNCTION OF ORPHAN HUMAN CYTOCHROME P450S
Zhong-Liu Wu, Katarina Stark, Zhong-Mei Tang, S. Giovana Salamanca-Pin ...
Session ID: S2-3
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.17.0
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(423K)
SAFROLE AND HUMAN CYTOCHROME P450: BIOACTIVATION, INHIBITION, AND INDUCTION
Yune-Fang Ueng
Session ID: S2-4
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.18.0
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(363K)
CYP3A5, GENDER, AND INTESTINAL ENZYME EXPRESSION AFFECT PHARMACOKINETICS OF NIFEDIPINE
Jin-ding Huang
Session ID: S2-5
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.19.0
CONFERENCE PROCEEDINGS
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(332K)
Symposium 3
Transporter as the Cause of Disease and the Target of Pharmacotherapy
IDENTIFICATION OF ABCG2/BCRP AS A MAJOR CAUSE FOR GOUT
Hirotaka Matsuo, Tappei Takada, Kimiyoshi Ichida, Hiroshi Suzuki, Nari ...
Session ID: S3-1
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.20.0
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(377K)
DISCOVERY AND IDENTIFICATION OF NOVEL DRUG TARGETS BASED ON THE ANALYSIS OF THE EXPRESSION AND FUNCTION OF DISEASE-ASSOCIATED ABC TRANSPORTERS
Tsuyoshi Shuto
Session ID: S3-2
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.21.0
CONFERENCE PROCEEDINGS
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(366K)
NPC1L1, A PHARMACOLOGICAL TARGET OF DYSLIPIDEMIA
Tappei Takada, Yoshihide Yamanashi, Hiroshi Suzuki
Session ID: S3-3
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.22.0
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(357K)
RESEARCH ON TRANSPORTERS IN DRUG DISCOVERY AND DEVELOPMENT
Noriko Okudaira
Session ID: S3-4
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.23.0
CONFERENCE PROCEEDINGS
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(371K)
Symposium 4
Fundamentals and Prospects of UDP-glucuronyltransferase (UGT) in Drug Development
New Aspects of UDP-glucuronosyltransferase
Hiroshi Yokota
Session ID: S4-1
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.24.0
CONFERENCE PROCEEDINGS
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(392K)
TRANSCRIPTIONAL REGULATION OF HUMAN UDP-GLUCURONOSYLTRANSFERASE UGT1A1 GENE EXPRESSION AND THE ALTERATION IN ITS PROTEIN EXPRESSION BY INTRACELLULAR FACTORS CONTROLLING CELL PROLIFERATION
Junko Sugatani
Session ID: S4-2
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.25.0
CONFERENCE PROCEEDINGS
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(358K)
DEVELOPMENT OF GLUCURONIDE PREPARATION SYSTEM FOR XENOBIOTIC METABOLITES USING GENETICALLY ENGINEERED BUDDING YEAST
Shinichi Ikushiro, Toshiyuki Sakaki
Session ID: S4-3
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.26.0
CONFERENCE PROCEEDINGS
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(375K)
PROTEIN-PROTEIN ASSOCIATION OF CYTOCHROME P450 AND UDP-GLUCURONOSYLTRANSFERASE: ITS RELEVANCE TO ENZYME FUNCTION
Yuji Ishii
Session ID: S4-4
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.27.0
CONFERENCE PROCEEDINGS
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(377K)
EVALUATION OF IN VITRO GLUCURONIDATION
Miki Nakajima
Session ID: S4-5
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.28.0
CONFERENCE PROCEEDINGS
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(366K)
Round Table 1
Chemically Reactive Drug Metabolites in Drug Discovery and Development
STRATEGY FOR PREDICTION OF DRUG-DRUG INTERACTIONS CAUSED BY MECHANISM-BASED INHIBITION IN THE DRUG DISCOVERY THROUGH DEVELOPMENT STAGES
Nobuo Sekiguchi, Motohiro Kato, Atsuko Higashida, Shotaro Takata, Masa ...
Session ID: R1-1
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.29.0
CONFERENCE PROCEEDINGS
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(353K)
CHRACTERIZATION OF REACTIVE METABOLITES BY HIGH-RESOLUTION MASS SPECTROMETRY IN DRUG DISCOVERY
Tomoyuki Ohe
Session ID: R1-2
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.30.0
CONFERENCE PROCEEDINGS
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(388K)
A ZONE CLASSIFICATION SYSTEM FOR RISK ASSESSMENT OF IDIOSYNCRATIC DRUG TOXICITY USING DAILY DOSE AND COVALENT BINDING
Shintaro Nakayama, Ryo Atsumi, Hideo Takakusa, Yoshimasa Kobayashi, At ...
Session ID: R1-3
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.31.0
CONFERENCE PROCEEDINGS
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(377K)
APPROACHES TO PREDICT IDIOSYNCRATIC AND IMMUNE-MEDIATED DRUG-INDUCED LIVER INJURY
Tsuyoshi Yokoi
Session ID: R1-4
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.32.0
CONFERENCE PROCEEDINGS
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(358K)
Round Table 2
The Significance and Issues of Evaluating Intestinal Metabolism in Drug Discovery and Development - Focused on CYP and UGT
CYP AND UGT EXPRESSED IN INTESTINE AND THEIR SPECIES DIFFERENCES
Miki Nakajima
Session ID: R2-1
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.33.0
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(360K)
QUANTITATIVE ASSESSMENT OF SMALL INTESTINAL METABOLSIM: CURRENT STATE AND ISSUES
Takashi Mizuma
Session ID: R2-2
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.34.0
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THE IMPACT OF INTESTINAL GLUCURONIDATION ON THE PHARMACOKINETICS OF RALOXIFENE IN RATS
Keigo Kosaka
Session ID: R2-3
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.35.0
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(370K)
THE INTESTINAL METABOLISM IN HUMANS AND MONKEYS.
DOES MONKEY PREDICT HUMAN PK? OR JUST EVOLVED
Takafumi Akabane, Kenji Tabata, Keitaro Kadono, Shuuichi Sakuda, Shige ...
Session ID: R2-4
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.36.0
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ANIMAL MODELS FOR PREDICTING INTESTINAL METABOLISM OF DRUDS IN HUMANS
Jiro Kuze
Session ID: R2-5
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.37.0
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(363K)
Forum 2010
The Status and Future Perspective of Protein Drugs: Their Safety, Pharmacokinetics and Approval
GLOBAL/DOMESTIC MARKET AND DEVELOPMENT STATUS OF BIOLOGICS
Eiji Takahara
Session ID: F1
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.38.0
CONFERENCE PROCEEDINGS
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(407K)
REGULATORY CMC ISSUES OF PROTEIN DRUGS
Koji Kawakami
Session ID: F2
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.39.0
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(436K)
Quality and Safety Evaluation of Biotechnology-Derived Pharmaceuticals
Toru Kawanishi
Session ID: F3
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.40.0
CONFERENCE PROCEEDINGS
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(383K)
THE IMPACT OF CLINICALPHARMACOLOGY APPROACHES IN MONOCLONAL ANTIBODY DEVELOPMENT
Kimio Terao
Session ID: F4
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.41.0
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(412K)
PHARMACOKINETIC STUDIES OF PROTEIN, PEPTIDE AND ANTIBODY DRUGS -REGULATIONS AND OPERATIONS-
Takuo Ogihara
Session ID: F5
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.42.0
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(405K)
CLINICAL TRIALS FOR DEVELOPMENTS OF BIOLOGIC DRUGS SUCH AS PROTEINS, PEPTIDES AND ANTIBODIES
Yuji Kumagai
Session ID: F6
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.43.0
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(405K)
Oral Presentations 1. Transporter - 1
UREMIC TOXIN TRANSPORTER SLCO4C1 IS ENHANCED BY STATINS
Takehiro Suzuki, Takahumi Toyohara, Yasutoshi Akiyama, Yoichi Takuuchi ...
Session ID: 1-C-9-1
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.44.0
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(335K)
INVOLVEMENT OF NOVEL HUMAN RIBOFLAVIN TRANSPORTERS hRFTs IN RIBOFLAVIN UPTAKE BY INTESTINAL T84 CELLS
Hiroki Yoshimatsu, Atsushi Yonezawa, Yoshiaki Yao, Satohiro Masuda, To ...
Session ID: 1-C-9-2
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.45.0
CONFERENCE PROCEEDINGS
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(335K)
ROLE OF GABA TRANSPORTER IN THE HEPATIC UPTAKE OF GUANIDINOACETATE
Masanori Tachikawa, Jun Fujinawa, Saori Ikeda, Shin-ichi Akanuma, Ken- ...
Session ID: 1-C-9-3
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.46.0
CONFERENCE PROCEEDINGS
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(338K)
THE BLOOD-TO-LIVER TRANSPORT OF TAURINE
Saori Ikeda, Shin-ichi Akanuma, Masanori Tachikawa, Ken-ichi Hosoya
Session ID: 1-C-9-4
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.47.0
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(338K)
EFFECT OF TICLOPIDINE ON MDR3/ABCB4-MEDIATED BILIARY SECRETION OF PHOSPHOLIPIDS
Takashi Yoshikado, Tappei Takada, Kousei Ito, Tomofumi Santa, Hiroshi ...
Session ID: 1-C-9-5
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.48.0
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(335K)
Oral Presentations 2. Transporter - 2
CALPAIN-MEDIATED CLEAVAGE NEGATIVELY REGULATES THE EXPRESSION LEVEL OF ABCG1
Natsuki Hori, Hisamitsu Hayashi, Yuichi Sugiyama
Session ID: 1-C-10-1
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.49.0
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DIFFERENTIAL EXPRESSION OF ORGANIC CATION TRANSPORTERS IN RAT DORSAL ROOT GANGLIA
Nancy N Jong, Johnson J Liu, Mark J McKeage, Takeo Nakanishi, Ikumi Ta ...
Session ID: 1-C-10-2
Published: 2010
Released on J-STAGE: December 15, 2010
DOI
https://doi.org/10.14896/jssxmeeting.25.0.50.0
CONFERENCE PROCEEDINGS
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(337K)
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