The Journal of Antibiotics
Online ISSN : 1881-1469
Print ISSN : 0021-8820
ISSN-L : 0021-8820
ASPERLICIN, A NOVEL NON-PEPTIDAL CHOLECYSTOKININ ANTAGONIST FROM ASPERGILLUS ALLIACEUS
FERMENTATION, ISOLATION AND BIOLOGICAL PROPERTIES
M. A. GOETZM. LOPEZR. L. MONAGHANR. S. L. CHANGV. J. LOTTIT. B. CHEN
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1985 年 38 巻 12 号 p. 1633-1637

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The fermentation and isolation of a new, non-peptide cholecystokinin antagonist, asperlicin, produced by Aspergillus alliaceus is described. The potent and specific interaction of asperlicin with cholecystokinin receptors was shown using in vitro biochemical assays.

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© Japan Antibiotics Research Association
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