JAPANESE CIRCULATION JOURNAL
Online ISSN : 1347-4839
Print ISSN : 0047-1828
ISSN-L : 0047-1828
EFFECT OF SEVERAL PROTEINASE INHIBITORS ON RENIN REACTION
TATSUO KOKUBUKUNIO HIWADAYUKIO NAGASAKAYUICHI YAMAMURA
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ジャーナル フリー

1974 年 38 巻 11 号 p. 955-958

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抄録
Inhibitory effect of the following nine proteinase inhibitors on the renin activity was studied. These were four kinds of trypsin inhibitors, Trasylol, pepstatin A, chymostatin, antipain and leupeptin. Except pepstatin A, none of these inhibited renin in vitro. The type of inhibition of renin by pepstatin A was competitive. Ki value for pepstatin A was found to be 3.2 × 10-7M.
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© Japanese Circulation Society
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