Drug Discoveries & Therapeutics
Online ISSN : 1881-784X
Print ISSN : 1881-7831
ISSN-L : 1881-7831
Original Articles
A facile method for the synthesis of N-(α-aminoacyl) sulfonamides
Shaolei WuMinglu ChenYutao WangXuben HouXinying YangLi SuHao Fang
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2012 Volume 6 Issue 2 Pages 62-68

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Abstract

N-Acylsulfonamide derivatives have important applications in organic synthesis and drug discovery. It was found that many problems occurred preparing amino acid derived N-acylsulfonamides with the commonly used coupling approach in our previous studies. In this paper, we report an efficient approach to synthesize various amino acids derived N-acylsulfonamides in high yields without any racemization.

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© 2012 International Research and Cooperation Association for Bio & Socio-Sciences Advancement
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