Synthesis and Biological Activity of 1, 2-Dithiolanes and 1, 2-Dithianes Bearing a Nitrogen-containing Substituent

抄録

A series of 1, 2-dithiolanes, 1, 2-dithianes and related compounds bearing a nitrogen-containig substituent were synthesized and their pesticidal activity was tested. A new general synthetic route to 1, 2-dithiolanes was established from 1, 3-diols. A variation in the position and character of the nitrogen atom is shown to be allowable to some extent for promoting insecticidal activity, unlike the case of sulfur atoms. Most compounds showed acaricidal activity, the strongest being displayed by cis-3, 5-bis (dimethylaminomethyl)-1, 2-dithiolane.