パラジウム触媒不斉アリルアミノ化反応を利用した CP-99,994 およびL-733,061の合成　

抄録

We developed the new S,O- and N,N-acetal type chiral ligands. Moreover we demonstrated both the catalytic asymmetric synthesis of (-)-CP-99,994 and (-)-L-733,061 using Pd-catalyzed asymmetric allylic amination as a key step.

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