著者所属：Department of Pharmaceutical Science, National Institute of Radiological Sciences Department of Pharmaceutical Science, National Institute of Radiological Sciences Department of Pharmaceutical Science, National Institute of Radiological Sciences Department of Pharmaceutical Science, National Institute of Radiological Sciences
Ten kinds of N-substituted-2-(2-aminoethyl)thiopseudoureas (AETs) were prepared. 1'-Phenyl-AET (VI) gave 2-aminothiazoline derivative (XXIII) with one equivalent of alkali, while other AETs having at least one hydrogen atom at the amino nitrogen underwent intramolecular rearrangement to give MEGs. GEDs were prepared from these MEGs by mild oxidation. The NMR and IR spectra of these compounds were also discussed.
